| Assay ID | Title | Year | Journal | Article |
|---|
| AID640180 | Displacement of [3H]bungarotoxin from nAChR alpha7 receptor on rat cortical membrane homogenate by gamma-counting | 2012 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 22, Issue:2
| Synthesis and binding affinity at α4β2 and α7 nicotinic acetylcholine receptors of new analogs of epibatidine and epiboxidine containing the 7-azabicyclo[2.2.1]hept-2-ene ring system. |
| AID361550 | Displacement of [125I]alpha-bungarotoxin from alpha7 nAChR in Wistar rat hindlimb muscle | 2008 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 18, Issue:16
| Epiboxidine and novel-related analogues: a convenient synthetic approach and estimation of their affinity at neuronal nicotinic acetylcholine receptor subtypes. |
| AID640182 | Displacement of [3H]methyllycaconitine from nAChR alpha7 receptor | 2012 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 22, Issue:2
| Synthesis and binding affinity at α4β2 and α7 nicotinic acetylcholine receptors of new analogs of epibatidine and epiboxidine containing the 7-azabicyclo[2.2.1]hept-2-ene ring system. |
| AID640185 | Selectivity ratio of Ki for displacement of [3H]nicotine from nAChR alpha4beta2 receptor to Ki for displacement of [3H]methyllycaconitine from nAChR alpha7 receptor | 2012 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 22, Issue:2
| Synthesis and binding affinity at α4β2 and α7 nicotinic acetylcholine receptors of new analogs of epibatidine and epiboxidine containing the 7-azabicyclo[2.2.1]hept-2-ene ring system. |
| AID146937 | Binding affinity towards Nicotinic acetylcholine receptor alpha-7 using [3H]-MLA as radioligand | 2003 | Bioorganic & medicinal chemistry letters, Sep-01, Volume: 13, Issue:17
| Synthesis and nicotinic binding of novel phenyl derivatives of UB-165. Identifying factors associated with alpha7 selectivity. |
| AID361553 | Selectivity ratio of Ki for rat alpha4beta2 nAChR to Ki for rat alpha7 nAChR | 2008 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 18, Issue:16
| Epiboxidine and novel-related analogues: a convenient synthetic approach and estimation of their affinity at neuronal nicotinic acetylcholine receptor subtypes. |
| AID640181 | Displacement of [3H]nicotine from nAChR alpha4beta2 receptor | 2012 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 22, Issue:2
| Synthesis and binding affinity at α4β2 and α7 nicotinic acetylcholine receptors of new analogs of epibatidine and epiboxidine containing the 7-azabicyclo[2.2.1]hept-2-ene ring system. |
| AID3056 | In vitro binding affinity towards (alpha-4)2(beta-2)3 neuronal nicotinic acetylcholine receptor in P2 membrane fractions of rat forebrain | 2003 | Journal of medicinal chemistry, May-22, Volume: 46, Issue:11
| 3D QSAR analyses-guided rational design of novel ligands for the (alpha4)2(beta2)3 nicotinic acetylcholine receptor. |
| AID146004 | Binding affinity towards alpha3-beta4 subtype of neuronal nicotinic acetylcholine receptor (nAChR) using [3H]epibatidine as radioligand | 2003 | Bioorganic & medicinal chemistry letters, Sep-01, Volume: 13, Issue:17
| Synthesis and nicotinic binding of novel phenyl derivatives of UB-165. Identifying factors associated with alpha7 selectivity. |
| AID640186 | Selectivity ratio of Ki for displacement of [3H]epibatidine from nAChR alpha4beta2 receptor to Ki for displacement of [3H]methyllycaconitine from nAChR alpha7 receptor | 2012 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 22, Issue:2
| Synthesis and binding affinity at α4β2 and α7 nicotinic acetylcholine receptors of new analogs of epibatidine and epiboxidine containing the 7-azabicyclo[2.2.1]hept-2-ene ring system. |
| AID146471 | Binding affinity towards Nicotinic acetylcholine receptor alpha4-beta2 using [3H]nicotine as radioligand | 2003 | Bioorganic & medicinal chemistry letters, Sep-01, Volume: 13, Issue:17
| Synthesis and nicotinic binding of novel phenyl derivatives of UB-165. Identifying factors associated with alpha7 selectivity. |
| AID465084 | Selectivity of beta4 nAChR over beta2 nAChR | 2010 | Journal of natural products, Mar-26, Volume: 73, Issue:3
| Phantasmidine: an epibatidine congener from the ecuadorian poison frog Epipedobates anthonyi. |
| AID361548 | Displacement of [3H]nicotine from alpha4beta2 nAChR in rat brain membrane | 2008 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 18, Issue:16
| Epiboxidine and novel-related analogues: a convenient synthetic approach and estimation of their affinity at neuronal nicotinic acetylcholine receptor subtypes. |
| AID640179 | Displacement of [3H]epibatidine from nAChR alpha4beta2 receptor on rat cortical membrane homogenate by beta-counting | 2012 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 22, Issue:2
| Synthesis and binding affinity at α4β2 and α7 nicotinic acetylcholine receptors of new analogs of epibatidine and epiboxidine containing the 7-azabicyclo[2.2.1]hept-2-ene ring system. |
| AID640183 | Displacement of [3H]epibatidine from nAChR alpha4beta2 receptor | 2012 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 22, Issue:2
| Synthesis and binding affinity at α4β2 and α7 nicotinic acetylcholine receptors of new analogs of epibatidine and epiboxidine containing the 7-azabicyclo[2.2.1]hept-2-ene ring system. |
| AID361549 | Displacement of [125I]alpha-bungarotoxin from alpha7 nAChR in rat brain membrane | 2008 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 18, Issue:16
| Epiboxidine and novel-related analogues: a convenient synthetic approach and estimation of their affinity at neuronal nicotinic acetylcholine receptor subtypes. |
| AID640184 | Selectivity ratio of Ki for displacement of [3H]epibatidine from nAChR alpha4beta2 receptor on rat cortical membrane homogenate to Ki for displacement of [3H]bungarotoxin from nAChR alpha7 receptor on rat cortical membrane homogenate | 2012 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 22, Issue:2
| Synthesis and binding affinity at α4β2 and α7 nicotinic acetylcholine receptors of new analogs of epibatidine and epiboxidine containing the 7-azabicyclo[2.2.1]hept-2-ene ring system. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |